Letters in Drug Design & Discovery

Author(s): Jianjun Shi, Guihua Ren, Zhimeng Dai, Ningjie Wu, Jianquan Weng, Tianming Xu, Xinghai Liu* and Chengxia Tan*

DOI: 10.2174/1570180814666170505123102

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Synthesis and Herbicidal Evaluation of Aryloxyphenoxypropionate Derivatives Containing Purine Moiety

Page: [15 - 20] Pages: 6

  • * (Excluding Mailing and Handling)

Abstract

Background: A series of purinoxyphenoxypropionates were designed and synthesized by introducing 8-(trifluoromethyl)-9H-purine into the aryloxyphenoxypropionate backbone.

Methods: The products were characterized by 1H NMR and HRMS.

Results and Conclusion: Preliminary bioassays indicated that most of the compounds exhibited good herbicidal activity at 200 mg/L.

Keywords: Purinoxyphenoxypropionates, herbicidal activity, ACCase, synthesis, antimycobacterial, antiviral.