Search Result "Falcipain-2"


Mini-Review Article
Falcipain-2 and Falcipain-3 Inhibitors as Promising Antimalarial Agents

Journal: Current Medicinal Chemistry

Volume: 28 Issue: 1 Year: 2021 Page: 3037-3058

Author(s): Roberta Ettari,Santo Previti,Carla Di Chio,Maria Zappalà

Design, Synthesis and Preliminary Screening of Some New Conformationally Constrained Falcipain-2 Inhibitors as Potential Antimalarial Agents

Journal: Letters in Drug Design & Discovery

Volume: 6 Issue: 4 Year: 2009 Page: 258-267

Author(s): Anil K. Shinde, Bishram S. Chouhan, Shirshendu Dasgupta, Rajani Giridhar, Philip Rosenthal, Jiri Gut, Mange R. Yadav

Profiling the Structural Determinants of Heteroarylnitrile Scaffold-Based Derivatives as Falcipain-2 Inhibitors by In Silico Methods

Journal: Current Medicinal Chemistry

Volume: 20 Issue: 1 Year: 2013 Page: 2032-2042

Author(s): Jinghui Wang, Yan Li, Yinfeng Yang, Shuwei Zhang, Ling Yang

Research Article
Combined CADD and Virtual Screening to Identify Novel Nonpeptidic Falcipain-2 Inhibitors

Journal: Current Computer-Aided Drug Design

Volume: 17 Issue: 4 Year: 2021 Page: 579-588

Author(s): Trisha Rajguru,Dipshikha Bora,Mahendra Kumar Modi

Oxidation and Tyrosine Nitration Induce Structural Changes and Inhibits Plasmodium falciparum Falcipain-2 Activity In Vitro

Journal: Protein & Peptide Letters

Volume: 23 Issue: 6 Year: 2016 Page: 562-572

Author(s): Jean B. Bertoldo,Hernán Terenzi

Research Article
Inhibition of Hemoglobin Degrading Protease Falcipain-2 as a Mechanism for Anti-Malarial Activity of Triazole-Amino Acid Hybrids

Journal: Current Topics in Medicinal Chemistry

Volume: 20 Issue: 5 Year: 2020 Page: 377-389

Author(s): Vigyasa Singh,Rahul Singh Hada,Amad Uddin,Babita Aneja,Mohammad Abid,Kailash C. Pandey,Shailja Singh

Falcipain Inhibition as a Promising Antimalarial Target

Journal: Current Topics in Medicinal Chemistry

Volume: 12 Issue: 5 Year: 2012 Page: 408-444

Author(s): Maria Marco, Jose Miguel Coteron

Cysteine Proteases of Malaria Parasites: Targets for Chemotherapy

Journal: Current Pharmaceutical Design

Volume: 8 Issue: 1 Year: 2002 Page: 1659-1672

Author(s): Philip J. Rosenthal, Puran S. Sijwali, Ajay Singh, Bhaskar R. Shenai

Review Article
Targeting Cysteine Proteases from Plasmodium falciparum: A General Overview, Rational Drug Design and Computational Approaches for Drug Discovery

Journal: Current Drug Targets

Volume: 19 Issue: 5 Year: 2018 Page: 501-526

Author(s): Boris D. Bekono,Fidele Ntie-Kang,Luc C. Owono Owono,Eugene Megnassan

Research Article
Synthesis, Antimalarial Evaluation and SAR Study of Some 1,3,5-Trisubstituted Pyrazoline Derivatives

Journal: Letters in Organic Chemistry

Volume: 16 Issue: 10 Year: 2019 Page: 807-817

Author(s): Shilpy Aggarwal,Deepika Paliwal,Dhirender Kaushik,Girish Kumar Gupta,Ajay Kumar

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