Search Result "Estrone sulfatase"


Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 8 Year: 2014 Page: 985-992
Author(s): Mohsen Akbarzadeh,Timothy Cartledge,Sabbir Ahmed

Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 3 Year: 2011 Page: 241-245
Author(s): Amit Kumar, Sukriti Singh, Hadi Bordbar, Timothy Cartledge, Sabbir Ahmed

Review of Estrone Sulfatase and its Inhibitors - An Important New Target Against Hormone Dependent Breast Cancer

Journal: Current Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2002 Page: 263-273
Author(s): Sabbir Ahmed, Caroline P. Owen, Karen James, Luther Sampson, Chirag K. Patel

Synthesis and In Vitro Biochemical Evaluation of a Series of Cycloalkyl Esters of 4-Sulfamoylated Benzoic Acid as Inhibitors of Estrone Sulfatase (ES)

Journal: Letters in Drug Design & Discovery
Volume: 4 Issue: 6 Year: 2007 Page: 399-403
Author(s): Caroline P. Owen, Chirag K. Patel, Tim Cartledge, Sabbir Ahmed

Estrone Sulfatase and Its Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 9 Issue: 6 Year: 2009 Page: 599-612
Author(s): Kwabina Aidoo-Gyamfi, Tim Cartledge, Kruti Shah, Sabbir Ahmed

Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 4 Year: 2014 Page: 437-443
Author(s): Sabbir Ahmed,Chirag K. Patel

Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 1 Year: 2011 Page: 26-31
Author(s): Chirag K. Patel, Sabbir Ahmed

Structure-Activity Relationship Determination Study of a Series of Novel Compounds as Potential Inhibitors of the Enzyme Estrone Sulfatase (ES)

Journal: Letters in Drug Design & Discovery
Volume: 1 Issue: 1 Year: 2004 Page: 35-44
Author(s): Chirag K. Patel, Caroline P. Owen, Kwabina Aidoo-Gyamfi, Sabbir Ahmed

Synthesis and In Vitro Biochemical Evaluation of a Series of Compounds as Potential Inhibitors of Estrone Sulfatase (ES) and the Role of pKa in both the Synthesis and the Inhibitory Activity of the Potential Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 4 Issue: 6 Year: 2007 Page: 394-398
Author(s): Caroline P. Owen, Mijal Patel, Chirag K Patel, Tim Cartledge, Sabbir Ahmed

In Vivo Inhibition of the Estrogen Sulfatase Enzyme and Growth of DMBA-Induced Mammary Tumors by Melatonin

Journal: Current Cancer Drug Targets
Volume: 10 Issue: 3 Year: 2010 Page: 279-286
Author(s): A. Gonzalez, V. Alvarez-Garcia, C. Martinez-Campa, M.D. Mediavilla, C. Alonso-Gonzalez, E.J. Sanchez-Barcelo, S. Cos

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