Search Result "CYP inactivation"


High Throughput Quantitative Assessment of CYP Inactivation Using 2 Concentration Points

Journal: Drug Metabolism Letters

Volume: 3 Issue: 2 Year: 2009 Page: 78-82

Author(s): Daniel Albaugh, Thomas Farrell, Michael Langan, W. George Lai

Assessment of Cytochrome P450 Enzyme Inhibition and Inactivation in Drug Discovery and Development

Journal: Current Topics in Medicinal Chemistry

Volume: 11 Issue: 4 Year: 2011 Page: 382-403

Author(s): David O. Nettleton, Heidi J. Einolf

Enzyme Kinetics for Clinically Relevant CYP Inhibition

Journal: Current Drug Metabolism

Volume: 6 Issue: 3 Year: 2005 Page: 241-257

Author(s): Zhi-Yi Zhang, Y. Nancy Wong

Altered CYP Expression and Function in Response to Dietary Factors: Potential Roles in Disease Pathogenesis

Journal: Current Drug Metabolism

Volume: 7 Issue: 1 Year: 2006 Page: 67-81

Author(s): Michael Murray

Assessment of the Inactivation Potential of Desethylamiodarone on Human CYP1A1

Journal: Drug Metabolism Letters

Volume: 4 Issue: 1 Year: 2010 Page: 9-14

Author(s): Marwa E. Elsherbiny, Ayman O.S. El-Kadi, Dion R. Brocks

Molecular Analysis and Modeling of Inactivation of Human CYP2D6 by Four Mechanism Based Inactivators

Journal: Drug Metabolism Letters

Volume: 6 Issue: 1 Year: 2012 Page: 7-14

Author(s): Mara Livezey, Leslie D. Nagy, Laura E. Diffenderfer, Evan J. Arthur, David J. Hsi, Jeffrey M. Holton, Laura Lowe Furge

CYP Inhibition-Mediated Drug-Drug Interactions

Journal: Current Enzyme Inhibition

Volume: 6 Issue: 3 Year: 2010 Page: 130-145

Author(s): Karoly Tihanyi, Monika L. Bakk, Eva Hellinger, Monika Vastag

cAMP-Mediated Regulation of CYP Enzymes and Its Application in Chemotherapy

Journal: Drug Metabolism Letters

Volume: 1 Issue: 3 Year: 2007 Page: 176-178

Author(s): Yoshihiro Ishikawa, Sayaka Suzuki, Koji Otsu, Coskun Ulucan, Kousaku Iwatsubo, Haruki Eguchi

Pharmacogenetic Variation in Drug Oxidizing CYPs: Impact on Drug Therapy, Drug Safety and Drug Interactions

Journal: Current Pharmacogenomics

Volume: 1 Issue: 3 Year: 2003 Page: 159-173

Author(s): Michael Murray

Research Article
Oxypeucedanin is a Mechanism-based Inactivator of CYP2B6 and CYP2D6

Journal: Current Drug Metabolism

Volume: 22 Issue: 11 Year: 2021 Page: 882-892

Author(s): Kehan Zhang,Yilin Li,Yao Fu,Tiantian Cui,Qian Wang,Xu Mao,Ying Peng,Jiang Zheng

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