Search Result "Bromodomain and extra-C terminal bromodomain inhibitors"


Research Article

Prediction of Inhibition Activity of BET Bromodomain Inhibitors using Grid Search-Based Extreme Learning Machine and Molecular Docking

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 11 Year: 2021 Page: 1039-1049
Author(s): Oluwatoba Emmanuel Oyeneyin,Babatunde Samuel Obadawo,Segun Michael Orimoloye,Eric Oluwafisayo Akintemi,Nureni Ipinloju,Adeola M. Asere,Taoreed O. Owolabi

Review Article

Privileged Scaffolds Targeting Bromodomain-containing Protein 4

Journal: Current Topics in Medicinal Chemistry
Volume: 22 Issue: 7 Year: 2022 Page: 600-627
Author(s):

Review Article

Bromodomain Protein-directed Agents and MYC in Small Cell LungCancer

Journal: Current Cancer Drug Targets
Volume: 24 Issue: 9 Year: 2024 Page: 930-940
Author(s):

Research Article

The Bromodomain and Extra-Terminal Protein Inhibitor OTX015 Suppresses T Helper Cell Proliferation and Differentiation

Journal: Current Molecular Medicine
Volume: 18 Issue: 9 Year: 2018 Page: 594-601
Author(s): Xiao Hu,Lauren P. Schewitz-Bowers,Philippa J. P. Lait,David A. Copland,Madeleine L. Stimpson,Jing Jing Li,Yizhi Liu,Andrew D. Dick,Richard W. J. Lee,Lai Wei

Research Article

Charting the Bromodomain BRD4: Towards the Identification of Novel Inhibitors with Molecular Similarity and Receptor Mapping

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 9 Year: 2018 Page: 1002-1011
Author(s): Fernando D. Prieto-Martinez,Jose L. Medina-Franco

Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 8 Year: 2015 Page: 776-794
Author(s): Lei Yu,Zhen Wang,Zhang Zhang,Xiaomei Ren,Xiaoyun Lu,Ke Ding

Review Article

Epigenetic Targets and their Inhibitors in Cancer Therapy

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 28 Year: 2018 Page: 2395-2419
Author(s): Le Zhao,Yong-Tao Duan,Ping Lu,Zhi-Juan Zhang,Xiao-Ke Zheng,Jun-Lei Wang,Wei-Sheng Feng

Review Article

BET Inhibitors as Anticancer Agents: A Patent Review

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 12 Issue: 4 Year: 2017 Page: 340-364
Author(s): Imran Ali,Gildon Choi,Kwangho Lee

Research Article

Piecing the Fragments Together: Dynamical Insights into the Enhancementof BRD4-BD1 (BET Protein) Druggability in Cancer ChemotherapyUsing Novel 8-methyl-pyrrolo[1,2-a]pyrazin-1(2H)-one Derivatives

Journal: Current Pharmaceutical Biotechnology
Volume: 23 Issue: 3 Year: 2022 Page: 444-456
Author(s): Oluwole B. Akawa,Opeyemi S. Soremekun,Fisayo A. Olotu,Mahmoud E.S. Solima

Current Frontiers

Targeting Protein-Protein Interaction with Covalent Small-Molecule Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 21 Year: 2019 Page: 1872-1876
Author(s): Bingbing Li,Deqin Rong,Yuanxiang Wang

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