Search Result "BRD4"

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Review Article
An Overview on Small Molecule Inhibitors of BRD4

Journal: Mini-Reviews in Medicinal Chemistry

Volume: 16 Issue: 17 Year: 2016 Page: 1403-1414

Author(s): Wenhai Huang,Xiaoliang Zheng,Yewei Yang,Xiaoju Wang,Zhengrong Shen

Research Article
Drug Discovery of Acetophenone Derivatives as BRD4 Inhibitors

Journal: Letters in Drug Design & Discovery

Volume: 17 Issue: 3 Year: 2020 Page: 323-329

Author(s): Zhimin Zhang,Wenhai Huang,Xiaoliang Zheng,Chuansheng Li,Zhengrong Shen

Review Article
Dual-target Inhibitors Based on BRD4: Novel Therapeutic Approaches for Cancer

Journal: Current Medicinal Chemistry

Volume: 28 Issue: 9 Year: 2021 Page: 1775-1795

Author(s): Sitao Zhang,Yanzhao Chen,Chengsen Tian,Yujing He,Zeru Tian,Yichao Wan,Tingting Liu

Mini-Review Article
BRD4 Protein as a Target for Lung Cancer and Hematological CancerTherapy: A Review

Journal: Current Drug Targets

Volume: 24 Issue: 14 Year: 2023 Page: 1079-1092

Author(s):

Research Article
Synthesis and Biological Activity of Quinoxalone Derivatives as BRD4 Bromodomain Inhibitors

Journal: Letters in Drug Design & Discovery

Volume: 14 Issue: 1 Year: 2017 Page: 50-57

Author(s): Bin Xu,Lei-Lei Zhao,Yi-Fei Yang,Jian Zhang,Ling-Yun Yang,Bing Zhang,Li Han,Hui-Bin Zhang,Jin-Pei Zhou

Research Article
Overexpression of BRD4 in Gastric Cancer and its Clinical Significance asa Novel Therapeutic Target

Journal: Current Cancer Drug Targets

Volume: 24 Issue: 2 Year: 2024 Page: 167-177

Author(s):

Research Article
Synthesis, Biological Evaluation and Molecular Docking Studies of Novel Trimethoxy-ring Derivatives as BRD4 Inhibitors

Journal: Letters in Drug Design & Discovery

Volume: 15 Issue: 1 Year: 2018 Page: 1319-1328

Author(s): Yan Yang,Zhiyi Yao

Research Article
The Klf6 Super-enhancer Determines Klf6 Sensitivity to BRD4 Inhibitors in Human Hepatoma (HepG2) Cells

Journal: Current Biotechnology

Volume: 9 Issue: 3 Year: 2020 Page: 209-218

Author(s): KumChol Ri,MyongRyong Ri,YongJae Song,KyuHwan Kim,Chol Kim

Twist-BRD4 Complex: Potential Drug Target for Basal-like Breast Cancer

Journal: Current Pharmaceutical Design

Volume: 21 Issue: 10 Year: 2015 Page: 1256-1261

Author(s): Jian Shi,Jingying Cao,Binhua P. Zhou

Research Article
Piecing the Fragments Together: Dynamical Insights into the Enhancementof BRD4-BD1 (BET Protein) Druggability in Cancer ChemotherapyUsing Novel 8-methyl-pyrrolo[1,2-a]pyrazin-1(2H)-one Derivatives

Journal: Current Pharmaceutical Biotechnology

Volume: 23 Issue: 3 Year: 2022 Page: 444-456

Author(s): Oluwole B. Akawa,Opeyemi S. Soremekun,Fisayo A. Olotu,Mahmoud E.S. Solima

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