Current Radiopharmaceuticals

Author(s): Johannes Ermert and Heinz H. Coenen

DOI: 10.2174/1874471011003020127

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No-Carrier-Added [18F]Fluorobenzene Derivatives as Intermediates for Built-up Radiosyntheses

Page: [127 - 160] Pages: 34

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Abstract

This review summarizes the possibilities of built-up syntheses of no-carrier-added radiofluorinated aromatic tracers via [18F]fluorobenzene derivatives as intermediate compounds.

Keywords: Fluorine-18, radiofluorination, nucleophilic substitution, built-up synthesis